Publications

[58] A decade of DNA-hybrid catalysis: from innovation to comprehension. Nicolas Duchemin, Isabelle Heath-Apostolopoulos, Michael Smietana,* Stellios Arseniyadis* Org. Biomol. Chem. 2017 (in press).

[57] Catalyse asymétrique innovante à base d’ADN. Stellios Arseniyadis,* Nicolas Duchemin, Isabelle Heath-Apostolopoulos, Michael Smietana* l’Actualité Chimique 2017 (in press).

[56] Radical Approaches in Natural Product Synthesis. Erica Benedetti, Cyril Bressy, Michael Smietana, Stellios Arseniyadis in Efficiency in Natural Products Total Synthesis, (Eds. P.-Q. Huang, Z.-J. Yao, R. P. Hsung), Wiley 2017 (in press).

[55] Multicomponent reactions in Natural Product Synthesis. Michael Smietana, Erica Benedetti, Cyril Bressy, Stellios Arseniyadis in Efficiency in Natural Products Total Synthesis, (Eds. P.-Q. Huang, Z.-J. Yao, R. P. Hsung), Wiley 2017 (in press).

[54] In situ targeted activation of a glucuronide prodrug using ultrasound-triggered release of composite droplets. Marine Bezagu, Jonathan Clarhaut, Brigitte Renoux, Fabrice Monti, Mickael Tanter, Patrick Tabeling,* Janine Cossy,* Olivier Couture, Sébastien Papot,* Stellios Arseniyadis* Eur. J. Med. Chem. 2017 (in press).

[53] A Pd-AAA approach to a-quaternary g-butyrolactones. Marllon Nascimento de Oliveira, Jeremy Fournier, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 201719, 14-17.

[52] Des produits naturels au développement d’outils synthétiques. Stellios Arseniyadis l’Actualité Chimique 2016, 413, 7-18.

[51] Total synthesis of putative 11-epi-lyngbouilloside aglycon. Amandine Kolleth, Julian Gebauer, Abdelatif ElMarrouni, Raphael Lebeuf, Céline Prévost, Eric Brohan, Stellios Arseniyadis,* Janine Cossy* Front. Chem. 20164, Article 34.

[50] Synthesis of Polyketides. Cyril Bressy, Michael Smietana, Erica Benedetti, Stellios Arseniyadis in From Biosynthesis to Total Synthesis, (Ed. A. L. Zografos), Wiley 2016 (in press).

[49] Expanding Biohybrid-mediated Asymmetric Catalysis into the Realm of RNA. Nicolas Duchemin, Erica Benedetti, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, Jean-Jacques Vasseur, Janine Cossy, Michael Smietana,* Stellios Arseniyadis* Chem. Commun201652, 8604-8607.

[48] Design, Synthesis and Binding Affinity Evaluation of Hoechst 33258 Derivatives for the Development of Sequence-specific DNA-based Asymmetric CatalystsKaren Amirbekyan, Nicolas Duchemin, Erica Benedetti, Rinah Joseph, Aude Colon, Shiraz A. Markarian, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, Janine Cossy, Jean-Jacques Vasseur, Stellios Arseniyadis,*  Michael Smietana* ACS Catal. 20166, 3096-3105.

[47] Selective Tsuji-Trost type C-allylation of hydrazones: A straightforward entry into 4,5-dihydro pyrazoles. Hachemia Elhachemia, Martin Cattoen, Marie Cordier, Janine Cossy, Stellios Arseniyadis, Hocine Ilitki*, Laurent El Kaïm* Chem. Commun201652, 14490-14493.

[46] A fast and switchable microfluidic mixer based on ultrasound-induced vaporization of perfluorocarbon. Marine Bezagu, Stellios Arseniyadis,* Janine Cossy,* Olivier Couture, Mickael Tanter, Fabrice Monti, Patrick Tabeling* Lab Chip 2015, 15, 2025-2029.

[45] DNA-cellulose: An economical, fully recyclable and highly effective chiral biomaterial for asymmetric catalysis. Erica Benedetti, Nicolas Duchemin, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, Jean-Jacques Vasseur, Janine Cossy, Michael Smietana,* Stellios Arseniyadis* Chem. Commun. 2015, 51, 6076-6079.

Supported DNA

[44] Recent Developments in Alkyne Borylations. Renaud Barberon, Erica Benedetti, Jean-Jacques Vasseur, Janine Cossy, Stellios Arseniyadis,* Michael Smietana,* Tetrahedron 201470, 8431-8452.

Metalloboration

[43] High spatiotemporal control of spontaneous reactions using ultrasound-triggered composite droplets. Marine Bezagu, Claudia Errico, Victor Chaulot-Talmon, Fabrice Monti, Mickael Tanter,  Patrick Tabeling,* Janine Cossy,*  Stellios Arseniyadis,*  Olivier Couture,   J. Am. Chem. Soc. 2014, 136, 7205-7208.

[42] Palladium-Catalyzed Allylic Alkylation of Allyl Dienol Carbonates: Reactivity, Regioselectivity, Enantioselectivity and Synthetic Applications. Stellios Arseniyadis,* Jérémy Fournier, Thangavelu Saravanan, Oscar Lozano, Sébastien Prevost, Alexis Archambeau, Candice Menozzi, Janine Cossy* Synlett 2013, 2350-2364. Special issue for the 5th Edition of the Young Investigator Workshop held in Marseille (invited article).

Synlett review

[41] DNA vs. Mirror Image DNA: A Universal Approach to Tune the Absolute Configuration in DNA-Based Asymmetric Catalysis. Jocelyn Wang, Erica Benedetti, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, Jean-Jacques Vasseur, Janine Cossy, Michael Smietana,* Stellios Arseniyadis* Angew. Chem. Int. Ed. 201352, 11546-11549.

L-DNA

[40] Non-enzymatic Acylative Kinetic Resolution of Primary Allylic Amines. Amandine Kolleth, Martin Cattoen, Stellios Arseniyadis,* Janine Cossy* Chem. Commun. 2013, 49, 9338-9340.

[39] Lyngbouilloside and Related Macrolides from Marine Cyanobacteria. Abdelatif ElMarrouni, Amandine Kolleth, Raphael Lebeuf, Julian Gebauer, Sébastien Prevost, Montserrat Heras, Stellios Arseniyadis,* Janine Cossy* Natural Product Communications 2013, 8, 965-972.

[38] Kinetic Resolution and Asymmetric Desymmetrization by Enantioselective Acylation and Related Processes. Alan C. Spivey,* Stellios Arseniyadis* in Comprehensive Enantioselective Organocatalysis, Ed. P. Dalko, Wiley-VCH 2013, Vol 3, Chapter 41, 1225-1284.

[37] Palladium-Catalyzed Asymmetric Allylic Alkylation of Cyclic Dienol Carbonates: Efficient Route to Enantioenriched g-Butenolides Bearing an All-Carbon a-Quaternary Stereogenic Center. Jeremy Fournier, Oscar Lozano, Candice Menozzi, Stellios Arseniyadis,* Janine Cossy* Angew. Chem. Int. Ed. 2013 52, 1257-1261 (Highlighted in Synfacts 2013, 4, 409).

[36] Kinetic Resolution of Propargylamines via a Highly Enantioselective Non-enzymatic N-Acylation Process. Amandine Kolleth, Sarah Christoph, Stellios Arseniyadis,* Janine Cossy* Chem. Commun. 2012, 48, 10511-10513.

[35] Catalysis-Based Enantioselective Total Synthesis of Myxothiazole Z, (14S)-Melithiazole G and (14S)‑Cystothiazole F. Aude Colon, Thomas J. Hoffman, Julian Gebauer, Jyotirmayee Dash, James H. Rigby, Stellios Arseniyadis,* Janine Cossy* Chem. Commun. 2012,48, 10508-10510.

[34] A Modular and Scalable One-pot Synthesis of Polysubstituted Furans. Jeremy Fournier, Stellios Arseniyadis,* Janine Cossy* Angew. Chem. Int. Ed. 2012, 51, 7562-7566.

[33] DNA as a Tool for Molecular Discovery. Michael Smietana,* Jean-Jacques Vasseur, Janine Cossy, Stellios Arseniyadis* in Modern Tools for the Synthesis of Complex Bioactive Molecules, (Eds.: J. Cossy, S. Arseniyadis), John Wiley & Sons, Inc., Hoboken, NJ, USA. 2012, 539-556.

[32] Total Synthesis of Nominal Lyngbouilloside Aglycon. Abdelatif ElMarrouni, Raphael Lebeuf, Julian Gebauer, Montserrat Heras, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2012, 14, 314-317.

[31] 2,6-bis[(4S)-4,5-Dihydro-4-(1-methylethyl)-5,5-diphenyl-2-oxazolyl] pyridine in electronic Encyclopedia of Organic Reagents (e-EROS), Wiley-VCH, 2011. Stellios Arseniyadis, Cyril Bressy.

[30] N-[(1S)-1-(Hydroxydiphenylmethyl)-3-methylbutyl]-2-pyrrolidinecarbox amide in electronic Encyclopedia of Organic Reagents (e-EROS), Wiley-VCH, 2011. Stellios Arseniyadis, Cyril Bressy.

[29] Studies Towards the N-Acylative Kinetic Resolution of NOBIN. Stellios Arseniyadis, Mohan Mahesh, Paul McDaid, Thomas Hampel, Stephen G. Davey, Alan C. Spivey* Coll. Czech. Chem. Commun. 2011, 76, 1239-1253.

[28] A Concise Approach towards the Synthesis of WS75624 A and WS75624 B via the cross-metathesis of vinyl-functionalized thiazoles. Jyotirmayee Dash, Bruno Melillo, Stellios Arseniyadis,* Janine Cossy* Tetrahedron Lett. 2011, 52, 2246-2249 (Special issue in honour of Professor Harry H. Wasserman on the occasion of his 90th birthday).

[27] Expedient Synthesis of a Stereoisomer of Acremolide B. Abdelatif ElMarrouni, Aya Fukuda, Montserrat Heras, Stellios Arseniyadis,* Janine Cossy* J. Org. Chem. 2010, 75, 8478-8486.

[26] Two Concise Total Syntheses of (-)-Bitungolide F. Abdelatif ElMarrouni, Shyamsunder R. Joolakanti, Aude Colon, Montserrat Heras, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2010, 12, 4074-4077.

[25] Stereoselective Synthesis of the C1‑C11 and C12‑C34 Fragments of Mycalolide A. Thomas J. Hoffman, Amandine Kolleth, James H. Rigby, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2010, 12, 3348-3351.

[24] Total Synthesis and Structural Revision of Vannusals A and B. Synthesis of the Originally Assigned Structure of Vannusal B. K. C. Nicolaou,* Adrian Ortiz, Hongjun Zhang, Philippe Dagneau, Andreas Lanver, Michael P. Jennings, Stellios Arseniyadis, Raffaella Faraoni, Dimitrios E. Lizos J. Am. Chem. Soc. 2010, 132, 7138-7152.

[23] Amine, Alcohol & Phosphine Catalysts for Acyl Transfer Reactions. Alan Spivey,* Stellios Arseniyadis* Topics in Current Chemistry: Asymmetric Organocatalysis, Ed. B. List, Springer Verlag 2010, Vol 291, Chapter 25, pp 233-280.

[22] Straightforward Synthesis of the Near-Infrared Fluorescent Voltage-Sensitive Dye RH1691 and Analogues thereof. Raphaël Lebeuf, Isabelle Férézou, Jean Rossier,Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2009, 11, 4822-4825.

[21] Enantioselective Organocatalytic Conjugate Reduction of b-Azole a,b‑Unsaturated Aldehydes. Thomas J. Hoffman, Jyotirmayee Dash, James H. Rigby, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2009, 11, 2756-2759.

[20] One-pot Hydrosilylation/RCM/Protodesilylation: Application to the Synthesis of w-Alkenyl a,b‑Unsaturated Lactones. Cyril Bressy, Frédéric Barggigia, Mathieu Guyonnet, Stellios Arseniyadis, Janine Cossy* Synlett, 2009, 565-568.

[19] Asymmetric Pentenylation of Aldehydes: A New Benchmark for the Preparation of Ethyl‑substituted Homoallylic Alcohols. Ravindra P. Sonawane, Shyamsunder R. Joolakanti, Stellios Arseniyadis,* Janine Cossy* Synlett 2009, 213-216.

[18] Asymmetric Total Synthesis of the Immunosuppressant (-)-Pironetin. Cyril Bressy, Jean-Pierre Vors, Stefan Hillebrand, Stellios Arseniyadis, Janine Cossy* Angew. Chem, Int. Ed. 2008, 47, 10137-10140.

[17] Formal Synthesis of Leustroducsin B. Joëlle Moïse, Ravindra P. Sonawane, Camilla Corsi, Sebastian V. Wendeborn, Stellios Arseniyadis,* Janine Cossy* Synlett 2008, 2617-2620.

[16] Total Synthesis of Cystothiazole A by Microwave-Assisted Olefin Cross-Metathesis. Julian Gebauer, Stellios Arseniyadis,* Janine Cossy* Eur. J. Org. Chem. 2008, 2701-2704.

[15] Synthesis of Vinyl-functionalized Oxazoles by Olefin Cross-Metathesis. Thomas J. Hoffman, James H. Rigby, Stellios Arseniyadis, Janine Cossy* J. Org. Chem. 2008, 73, 2400-2403.

[14] Facile Synthesis of the C1–C13 Fragment of Lyngbouilloside. Julian Gebauer, Stellios Arseniyadis,* Janine Cossy* Synlett 2008, 712-714.

[13] Non-enzymatic Kinetic Resolution of Amines in Ionic Liquids. Cyrille Sabot, Pithani V. Subhash, Alain Valleix, Stellios Arseniyadis,* Charles Mioskowski,* Synlett 2008, 268-272.

[12] A Concise Total Synthesis of Melithiazole C. Julian Gebauer, Stellios Arseniyadis, Janine Cossy* Org. Lett. 2007, 9, 3425-3427.

[11] The Chemistry and Biology of Epothilones – The Wheel keeps turning. Karl-Heinz Altmann,* Bernhard Pfeiffer, Stellios Arseniyadis, Benjamin A. Pratt, K. C. Nicolaou* ChemMedChem 2007, 396-423.

[10] Cross-Metathesis Between a‑Methylene-g-butyrolactone and Olefins: A Dramatic Additive Effect. Joëlle Moïse, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2007, 9, 1695-1698.

[9] Synthesis of Vinyl-Functionalized Thiazoles by Cross-Metathesis and Tandem Stille Coupling/Cross‑Metathesis. Jyotirmayee Dash, Stellios Arseniyadis, Janine Cossy* Adv. Synth. Cat. 2007, 349, 152-156.

[8] Molecular Design and Chemical Synthesis of a Highly Potent Epothilone. K. C. Nicolaou,* Benjamin A. Pratt, Stellios Arseniyadis, Markus Wartmann, Aurora O’Brate, Paraskevi Giannakakou ChemMedChem 2006, 1, 41-44.

[7] Rapid, Room-temperature Acylative Kinetic Resolution of sec-Alcohols using Atropisomeric 4‑Aminopyridine/triphenylphosphine Catalysis. Alan C. Spivey,* Stellios Arseniyadis, Tomasz Fekner, Adrian Maddaford, David P. Leese Tetrahedron 2006, 62, 295-301.

[6] Unprecedented, Fully Recyclable, Solid-Supported Reagent for the Kinetic Resolution of Racemic Amines through Enantioselective N‑Acetylation. Stellios Arseniyadis, Pithani V. Subhash, Alain Valleix, Alain Wagner,* Charles Mioskowski* Chem. Commun. 2005, 26, 3310-3312 (Highlighted in Synfacts 2005, 1, 170).

[5] Tuning the Enantioselective N-Acetylation of Racemic Amines: A Spectacular Salt Effect. Stellios Arseniyadis, Pithani V. Subhash, Alain Valleix, Suju P. Mathew,Donna G. Blackmond, Alain Wagner,* Charles Mioskowski* J. Am. Chem. Soc. 2005, 127, 6138-6139.

[4] Nucleophilic Catalysis by 4-(Dialkylamino)pyridines Revisited – The Search for Optimal Reactivity and Selectivity. Alan C. Spivey,* Stellios Arseniyadis Angew. Chem. Int. Ed. 2004, 43, 5436-5441.

[3] Kinetic Resolution of Amines: A Chemoselective and Highly Enantioselective Acetylating Agent with a Unique Solvent-induced Reversal of Stereoselectivity. Stellios Arseniyadis, Alain Valleix, Alain Wagner,* Charles Mioskowski* Angew. Chem. Int. Ed. 2004, 43, 3314-3317.

[2] Resin Bound 4-Phenyl-1,2-dihydroquinoline (DHQ): an New Safety-Catch Linker for Solid Phase Organic Synthesis (SPOS). Stellios Arseniyadis, Alain Wagner,* Charles Mioskowski* Tetrahedron Lett. 2004, 45, 2251-2253.

[1] A Straightforward Preparation of Amino-polystyrene Resin from Merrifield Resin. Stellios Arseniyadis, Alain Wagner,* Charles Mioskowski* Tetrahedron Lett. 2002, 43, 9717-9719.

 

Patent

Chemical synthesis of a highly potent epothilone. Nicolaou, K. C.; Pratt, B.; Arseniyadis, S. (International publication number: WO 2007/062288 International publication date: 31/05/2007).

Books

[2] Modern Tools for the Synthesis of Complex Bioactive Molecules. Janine Cossy, Stellios Arseniyadis, John Wiley & Sons, Inc., Hoboken, NJ, USA (2012), ISBN-13: 978-0470616185.

[1] Metathesis in Natural Product Synthesis. Janine Cossy, Stellios Arseniyadis, Christophe Meyer, Wiley-VCH, Weinheim, Germany (2010), ISBN-13: 978-3-527-32440-8.