[95] Collective synthesis of butenolide-containing mono-terpenoid natural products. Thomas Keenan, François Richard, Sidonie Aubert, Kelly Maurent, Alexandre Jean, Andrei Corbu,* Stellios Arseniyadis* (in preparation).

[94] A quest for selectivity in the Friedel-Crafts alkylation/enantioselective protonation using DNA-RNA hybrids. Sidonie Aubert, Nicolas Duchemin, João V. de Souza, Lucas Bethge, Stefan Vonhoff, Agnieszka K. Bronowska, Michael Smietana,* Stellios Arseniyadis* (in preparation).

[93] S-(Difluoromethyl)-S-phenyl-N-tosylsulfoxime: A highly effective and multifaceted difluoromethylating agent. Jinlei Zhang, Nicolas Duchemin, Shamim Fanai-Danesh, Nathan Long, Elias Selmi-Higashi, Stellios Arseniyadis* (in preparation).

[92] Photocatalysed bioinspired dimerization of piperine in batch and flow: [2+2] vs [4+2] under catalyst control. Amina Sesay, Mohammed Latrache, Jinlei Zhang, Samuel Oger, Stephen T. Hilton, Erwan Poupon, Stellios Arseniyadis* Laurent Evanno* (in preparation).

[91] Visible light-mediated difluoromethylation/cyclization in batch and flow: Scalable synthesis of CHF2-containing benzimidazo[2,1-a]isoquinolin-6(5H)-ones. Al Hannam, Phinyada Kankraisri, Karan R. Thombare, Prahallad Meher, Alexandre Jean, Stephen T. Hilton, Sandip Murarka,* Stellios Arseniyadis* (in preparation).

[90] Synthesis of CHF2-containing heterocycles through oxo-difluoromethylation using low-cost 3D-printed photoflow reactors. Jinlei Zhang, Elias Selmi-Higashi, Shen Zhang, Alexandre Jean, Stephen T. Hilton,* Xacobe C. Cambeiro,* and Stellios Arseniyadis* Org. Lett. 2024 (in press).

[89] Pd-Catalysed Asymmetric Allylic Alkylation of Heterocycles: A User’s Guide. François Richard, Paul Clark, Al Hannam, Thomas Keenan, Alexandre Jean, Stellios Arseniyadis* Chem. Soc. Rev. 2024 (in press).

[88] Chiral, air stable, and reliable Pd(0) precatalysts applicable to asymmetric allylic alkylation chemistry. Jingjun Huang, Thomas Keenan, Francois Richard, Jingru Lu, Sarah E. Jenny, Alexandre Jean, Stellios Arseniyadis,* David C. Leitch* Nat. Commun. 2023, 14, 8058. Open AccessChemRxiv 2023 (DOI: 10.26434/chemrxiv-2023-0xbh5).

[87] Palladium precatalyst embodiments for enantioselective chemical reactions and methods of making and using the same. David Leitch, Stellios Arseniyadis, Jingjun Huang (International publication number: WO2023156972A1, International publication date: 24/08/2023).

[86] Unlocking copper catalysis with nitro compounds: Synthesis of functionalized allylboranes from allylic nitroalkanes. Nicolas Fincias, Louis Clavier, Mansour Dole Kerim, Nicolas Casaretto, Julian Garrec, Stellios Arseniyadis,* Laurent. El Kaïm* ChemRxiv 2023 (DOI: 10.26434/chemrxiv-2023-mztk4).

[85] Late-stage functionalisation of pharmaceuticals, agrochemicals and natural products. François Richard, Elias Selmi-Higashi, Stellios Arseniyadis in Transition-metal-catalyzed C-H functionalization of heterocycles (Ed. T. Punniyamurthy and A. Kumar), Wiley & Sons (DOI: 10.1002/9781119774167.ch18).

[84] Expanding the 'aplysinospin cascade' through DNA-templated [2+2] photocycloaddition. Samuel Oger, Nicolas Duchemin, Mayssa Bendiab, Nicolas Birlirakis, Adam Skiredj, Somia Rharrabti, Remi Franco, Erwan Poupon,* Michael Smietana,* Stellios Arseniyadis,* Laurent Evanno* Chem. Commun. 2023, 59, 4221–4224. Open Access

[83] A new benchmark in DNA-based asymmetric catalysis: Prevalence of modified DNA/RNA hybrid systems. Nicolas Duchemin, Sidonie Aubert, João V. de Souza, Lucas Bethge, Stefan Vonhoff, Agnieszka K. Bronowska, Michael Smietana,* Stellios Arseniyadis* JACS Au 20222, 1910–1917. Open Access

[82] Enantioselective synthesis of γ-butenolides through Pd-catalysed C5-selective allylation of siloxyfurans. François Richard, Sidonie Aubert, Tania Katsina, Luuk Reinalda, David Palomas, Rachel Crespo-Otero, Jingjun Huang, David C. Leitch, Carlos Mateos, Stellios Arseniyadis* Nat. Synth. 2022, 1, 641–648.

[81] Phase-transfer catalyzed alkylation of hydantoins. Thomas Keenan, Alexandre Jean,* Stellios Arseniyadis* ACS Organic & Inorganic Au 2022, 2, 312317. Open Access

[80] DNA-based asymmetric catalysis: Past, present and future. Sidonie Aubert, Nicolas Duchemin, Jin-Lei Zhang, Michael Smietana, Stellios Arseniyadis* in Enantioselective Catalysis, Book series: Series on Chemistry, Energy and the Environment (Ed. A. Marinetti), World Scientific 2022 (DOI: 10.1142/9789811248436_0001).

[79] Four-membered rings with one sulfur and one nitrogen atom. François Richard, Jennifer Ciesielski, Stellios Arseniyadis in Comprehensive Heterocyclic Chemistry IV, (Ed. G. Evano), Elsevier 2021 (in press).

[78] Synthesis of α-difluoromethyl aryl ketones through a photoredox difluoromethylation of enol silanes. Elias Selmi-Higashi, Jinlei Zhang, Xacobe C. Cambeiro, Stellios Arseniyadis* Org. Lett. 2021, 23, 42394243.

[77] 4-Cyano-3-oxotetrahydrothiophene (c-THT): An ideal acrylonitrile anion equivalent. François Richard, Carlos Mateos, Stellios Arseniyadis* SynOpen 2021, 5, 25–28. Open Access

[76] O-Allylated Pudovik and Passerini adducts as versatile templates for product diversification. Mansour Dolé Kerim, Tania Katsina, Martin Cattoen, Nicolas Fincias, Stellios Arseniyadis,* Laurent El Kaïm* J. Org. Chem. 202085, 12514–12525.

[75] Direct access to highly enantioenriched α-branched acrylonitriles through a one-pot sequential asymmetric Michael addition/retro-Dieckmann/retro-Michael fragmentation cascade. Nicolas Duchemin, Martin Cattoen, Oscar Gayraud, Silvia Anselmi, Bilal Siddiq, Roberto Buccafusca, Marc Daumas, Vincent Ferey, Michael Smietana, Stellios Arseniyadis* Org. Lett. 2020, 22, 5995-6000.

  • ChemRxiv. 2020 (DOI: 10.26434/chemrxiv.12185535.v1)

[74] Aerobic oxidation of alcohols using catalytic DDQ/HNO3. Tania Katsina, Louis Clavier, Jean-François Giffard, Nayane Macedo Portela da Silva, Jean Fournier, Chloé Copin, Stellios Arseniyadis,* Alexandre Jean* Org. Process Res. Dev. 2020, 24, 856-860.

[73] DNA-based asymmetric inverse electron-demand hetero-Diels-Alder. Justine Mansot, Jimmy Lauberteaux, Aurélien Lebrun, Marc Mauduit, Jean-Jacques Vasseur, Renata Marcia de Figueiredo, Stellios Arseniyadis,* Jean-Marc Campagne,* Michael Smietana* Chem. Eur. J. 2020, 26, 35193523.

[72] A Sequential palladium‑catalyzed allylic alkylation/retro-Dieckmann fragmentation strategy for the synthesis of α-substituted acrylonitriles. Tania Katsina, Sachi Sharma, Roberto Buccafusca, Derek J. Quinn, Thomas S. Moody, Stellios Arseniyadis* Org. Lett201921, 9348–9352.

[71] Spatial and temporal control of chemical processes. Sidonie Aubert, Marine Bezagu, Alan C. Spivey,* Stellios Arseniyadis* Nature Rev. Chem. 20193, 706–722.

[70] A unified strategy for the synthesis of difluoromethyl- and vinylfluoride-containing scaffolds. Nicolas Duchemin, Roberto Buccafusca, Marc Daumas, Vincent Ferey, Stellios Arseniyadis* Org. Lett. 2019, 21, 82058210.

  • ChemRxiv 2019 (DOI: 10.26434/chemrxiv.8091314.v1)
  • Highlighted in OPR&D.

[69] A rational quest for selectivity through precise ligand-positioning in the tandem DNA-catalysed Friedel-Crafts alkylation/asymmetric protonation. Justine Mansot, Sidonie Aubert, Nicolas Duchemin, Jean-Jacques Vasseur, Stellios Arseniyadis,* Michael Smietana* Chem. Sci. 2019, 10, 28752881.

[68] A sequential Pd-AAA/CM/Cope rearrangement strategy for the stereoselective synthesis of γ-butenolides. Sidonie Aubert, Tania Katsina, Stellios Arseniyadis* Org. Lett. 2019, 21 , 22312235.

[67] Asymmetric synthesis of α-quaternary γ-lactams through palladium-catalyzed asymmetric allylic alkylation. Tao Song, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2019, 21, 603607.

[66] α,β-Unsaturated 2-acyl-imidazoles in asymmetric biohybrid catalysis. Justine Mansot, Jean-Jacques Vasseur, Stellios Arseniyadis,* Michael Smietana* ChemCatChem. 2019, 11, 5686–5704.

[65] DNA-templated [2+2] photocycloaddition: A straightforward entry into the aplysinopsin family of natural products. Nicolas Duchemin, Adam Skiredj, Justine Mansot, Karine Leblanc, Jean-Jacques Vasseur, Mehdi A. Beniddir, Laurent Evanno,* Erwan Poupon,* Michael Smietana,* Stellios Arseniyadis* Angew. Chem. Int. Ed. 2018, 57, 1178611791. Highlighted in Nature Reviews Chemistry and in the CNRS website.

[64] Challenges and opportunities in DNA-based asymmetric catalysis. Michael Smietana,* Stellios Arseniyadis* Chimia 2018, 72630634 - invited article.

[63] Highly enantioselective, base-free synthesis of α-quaternary succinimides through catalytic asymmetric allylic alkylation. Tao Song, Stellios Arseniyadis,* Janine Cossy* Chem. Eur. J. 2018, 24, 80768080 (selected as a Hot Paper). Highlighted in Synfact.

[62] Palladium-catalyzed asymmetric allylic alkylation of 4-substituted isoxazolidin-5-ones: A straightforward access to β2,2‑amino acids. Marllon Nascimento de Oliveira, Stellios Arseniyadis,* Janine Cossy* Chem. Eur. J. 201824, 48104814.

[61] Palladium-catalysed O-allylation of α-hydroxyphosphonates: An expedient entry into phosphono-oxaheterocycles. Mansour Dolé Kerim, Martin Cattoen, Nicolas Fincias, Aurélie Dos Santos, Stellios Arseniyadis,* Laurent El Kaïm* Adv. Synth. & Catal. 2018360, 449454 (selected as a Very Important Publication).

[60] Recent applications of Kagan's reagent (SmI2) in natural product synthesis. Erica Benedetti, Cyril Bressy, Michael Smietana, Stellios Arseniyadis in Efficiency in Natural Products Total Synthesis, (Eds. P.-Q. Huang, Z.-J. Yao, R. P. Hsung), Wiley 2018, ch 8, 319344.

[59] Multicomponent reactions in natural product synthesis. Michael Smietana, Erica Benedetti, Cyril Bressy, Stellios Arseniyadis in Efficiency in Natural Products Total Synthesis, (Eds. P.-Q. Huang, Z.-J. Yao, R. P. Hsung), Wiley 2018, ch 6, 273295.

[58] Dinucleating Schiff base ligand in Zn/4f coordination chemistry: Synthetic challenges and catalytic activity evaluation. Stavroula I. Sampani, Sidonie Aubert, Martin Cattoen, Kieran Griffiths, Alaa Abdul-Sada, Geoffrey R. Akien, Graham J. Tizzard, Simon J. Coles, Stellios Arseniyadis,* George E. Kostakis* Dalton Trans. 2018, 47, 44864493.

[57] A decade of DNA-hybrid catalysis: from innovation to comprehension. Nicolas Duchemin, Isabelle Heath-Apostolopoulos, Michael Smietana,* Stellios Arseniyadis* Org. Biomol. Chem. 2017, 15, 70727087.

[56] In situ targeted activation of a glucuronide prodrug using ultrasound-triggered release of composite droplets. Marine Bezagu, Jonathan Clarhaut, Brigitte Renoux, Fabrice Monti, Mickael Tanter, Patrick Tabeling,* Janine Cossy,* Olivier Couture, Sébastien Papot,* Stellios Arseniyadis* Eur. J. Med. Chem. 2017142, 27.

Image 1

[55] A Pd-AAA approach to a-quaternary g-butyrolactones. Marllon Nascimento de Oliveira, Jeremy Fournier, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 201719, 1417.

[54] Catalyse asymétrique innovante à base d’ADN. Stellios Arseniyadis,* Nicolas Duchemin, Isabelle Heath-Apostolopoulos, Michael Smietana* l'Actualité Chimique 2017, 417, 1727.

[53] Des produits naturels au développement d’outils synthétiques. Stellios Arseniyadis l'Actualité Chimique 2016, 413, 718.

[52] Total synthesis of putative 11-epi-lyngbouilloside aglycon. Amandine Kolleth, Julian Gebauer, Abdelatif ElMarrouni, Raphael Lebeuf, Céline Prévost, Eric Brohan, Stellios Arseniyadis,* Janine Cossy* Front. Chem. 20164, Article 34.

[51] Synthesis of polyketides. Cyril Bressy, Michael Smietana, Erica Benedetti, Stellios Arseniyadis in From Biosynthesis to Total Synthesis, (Ed. A. L. Zografos), Wiley 2016, ch 2, 19129.

[50] Expanding biohybrid-mediated asymmetric catalysis into the realm of RNA. Nicolas Duchemin, Erica Benedetti, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, Jean-Jacques Vasseur, Janine Cossy, Michael Smietana,* Stellios Arseniyadis* Chem. Commun201652, 86048607.

[49] Design, synthesis and binding affinity evaluation of Hoechst 33258 derivatives for the development of sequence-specific DNA-based asymmetric catalystsKaren Amirbekyan, Nicolas Duchemin, Erica Benedetti, Rinah Joseph, Aude Colon, Shiraz A. Markarian, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, Janine Cossy, Jean-Jacques Vasseur, Stellios Arseniyadis,* Michael Smietana* ACS Catal. 20166, 30963105.

[48] Selective Tsuji-Trost type C-allylation of hydrazones: A straightforward entry into 4,5-dihydro pyrazoles. Hachemia Elhachemia, Martin Cattoen, Marie Cordier, Janine Cossy, Stellios Arseniyadis, Hocine Ilitki*, Laurent El Kaïm* Chem. Commun201652, 1449014493.

[47] A fast and switchable microfluidic mixer based on ultrasound-induced vaporization of perfluorocarbon. Marine Bezagu, Stellios Arseniyadis,* Janine Cossy,* Olivier Couture, Mickael Tanter, Fabrice Monti, Patrick Tabeling* Lab Chip 2015, 15, 20252029.

[46] DNA-cellulose: An economical, fully recyclable and highly effective chiral biomaterial for asymmetric catalysis. Erica Benedetti, Nicolas Duchemin, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, Jean-Jacques Vasseur, Janine Cossy, Michael Smietana,* Stellios Arseniyadis* Chem. Commun. 2015, 51, 60766079. Highlighted in Chemistry World and in the CNRS website.

Supported DNA

[45] Recent developments in alkyne borylations. Renaud Barberon, Erica Benedetti, Jean-Jacques Vasseur, Janine Cossy, Stellios Arseniyadis,* Michael Smietana,* Tetrahedron 201470, 84318452.

[44] High spatiotemporal control of spontaneous reactions using ultrasound-triggered composite droplets. Marine Bezagu, Claudia Errico, Victor Chaulot-Talmon, Fabrice Monti, Mickael Tanter, Patrick Tabeling,* Janine Cossy,* Stellios Arseniyadis,* Olivier Couture, J. Am. Chem. Soc. 2014, 136, 72057208. Highlighted in the CNRS website.

[43] Palladium-catalyzed allylic alkylation of allyl dienol carbonates: Reactivity, regioselectivity, enantioselectivity and synthetic applications. Stellios Arseniyadis,* Jérémy Fournier, Thangavelu Saravanan, Oscar Lozano, Sébastien Prevost, Alexis Archambeau, Candice Menozzi, Janine Cossy* Synlett 2013, 23502364. Special issue for the 5th Edition of the Young Investigator Workshop held in Marseille (invited article).

Synlett review

[42] DNA vs. mirror image DNA: A universal approach to tune the absolute configuration in DNA-based asymmetric catalysis. Jocelyn Wang, Erica Benedetti, Lucas Bethge, Stefan Vonhoff, Sven Klussmann, Jean-Jacques Vasseur, Janine Cossy, Michael Smietana,* Stellios Arseniyadis* Angew. Chem. Int. Ed. 201352, 1154611549. Highlighted in the CNRS website.


[41] Non-enzymatic acylative kinetic resolution of primary allylic amines. Amandine Kolleth, Martin Cattoen, Stellios Arseniyadis,* Janine Cossy* Chem. Commun. 2013, 49, 93389340.

[40] Lyngbouilloside and related macrolides from marine cyanobacteria. Abdelatif ElMarrouni, Amandine Kolleth, Raphael Lebeuf, Julian Gebauer, Sébastien Prevost, Montserrat Heras, Stellios Arseniyadis,* Janine Cossy* Natural Product Communications 2013, 8, 965972.

[39] Regio‐ and position selective reactions and desymmetrizationsAlan C. Spivey,* Stellios Arseniyadis* in Comprehensive Enantioselective Organocatalysis, Ed. P. Dalko, Wiley-VCH 2013, Vol 3, Chapter 41, 12251284.

[38] Palladium-catalyzed asymmetric allylic alkylation of cyclic dienol carbonates: Efficient route to enantioenriched g-butenolides bearing an all-carbon a-quaternary stereogenic center. Jeremy Fournier, Oscar Lozano, Candice Menozzi, Stellios Arseniyadis,* Janine Cossy* Angew. Chem. Int. Ed. 2013 52, 12571261 (Highlighted in Synfacts 2013, 4, 409).

[37] Kinetic resolution of propargylamines via a highly enantioselective non-enzymatic N-acylation process. Amandine Kolleth, Sarah Christoph, Stellios Arseniyadis,* Janine Cossy* Chem. Commun. 2012, 48, 1051110513.

[36] Catalysis-based enantioselective total synthesis of myxothiazole Z, (14S)-melithiazole G and (14S)‑cystothiazole F. Aude Colon, Thomas J. Hoffman, Julian Gebauer, Jyotirmayee Dash, James H. Rigby, Stellios Arseniyadis,* Janine Cossy* Chem. Commun. 2012,48, 1050810510.

[35] A modular and scalable one-pot synthesis of polysubstituted furans. Jeremy Fournier, Stellios Arseniyadis,* Janine Cossy* Angew. Chem. Int. Ed. 2012, 51, 75627566.

[34] DNA as a tool for molecular discovery. Michael Smietana,* Jean-Jacques Vasseur, Janine Cossy, Stellios Arseniyadis* in Modern Tools for the Synthesis of Complex Bioactive Molecules, (Eds.: J. Cossy, S. Arseniyadis), John Wiley & Sons, Inc., Hoboken, NJ, USA. 2012, 539556.

[33] Total synthesis of nominal lyngbouilloside aglycon. Abdelatif ElMarrouni, Raphael Lebeuf, Julian Gebauer, Montserrat Heras, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2012, 14, 314317.

[32] 2,6-bis[(4S)-4,5-Dihydro-4-(1-methylethyl)-5,5-diphenyl-2-oxazolyl] pyridine in electronic Encyclopedia of Organic Reagents (e-EROS), Wiley-VCH, 2011. Stellios Arseniyadis, Cyril Bressy.

[31] N-[(1S)-1-(Hydroxydiphenylmethyl)-3-methylbutyl]-2-pyrrolidinecarbox amide in electronic Encyclopedia of Organic Reagents (e-EROS), Wiley-VCH, 2011. Stellios Arseniyadis, Cyril Bressy.

[30] Studies towards the N-acylative kinetic resolution of NOBIN. Stellios Arseniyadis, Mohan Mahesh, Paul McDaid, Thomas Hampel, Stephen G. Davey, Alan C. Spivey* Coll. Czech. Chem. Commun. 2011, 76, 12391253.

[29] A concise approach towards the synthesis of WS75624 A and WS75624 B via the cross-metathesis of vinyl-functionalized thiazoles. Jyotirmayee Dash, Bruno Melillo, Stellios Arseniyadis,* Janine Cossy* Tetrahedron Lett. 2011, 52, 22462249 (Special issue in honour of Professor Harry H. Wasserman on the occasion of his 90th birthday).

[28] Expedient synthesis of a stereoisomer of acremolide B. Abdelatif ElMarrouni, Aya Fukuda, Montserrat Heras, Stellios Arseniyadis,* Janine Cossy* J. Org. Chem. 2010, 75, 84788486.

[27] Two concise total syntheses of (-)-bitungolide F. Abdelatif ElMarrouni, Shyamsunder R. Joolakanti, Aude Colon, Montserrat Heras, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2010, 12, 40744077.

[26] Stereoselective synthesis of the C1‑C11 and C12‑C34 fragments of mycalolide A. Thomas J. Hoffman, Amandine Kolleth, James H. Rigby, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2010, 12, 33483351.

[25] Total synthesis and structural revision of vannusals A and B. Synthesis of the originally assigned structure of Vannusal B. K. C. Nicolaou,* Adrian Ortiz, Hongjun Zhang, Philippe Dagneau, Andreas Lanver, Michael P. Jennings, Stellios Arseniyadis, Raffaella Faraoni, Dimitrios E. Lizos J. Am. Chem. Soc. 2010, 132, 71387152.

[24] Amine, alcohol & phosphine catalysts for acyl transfer reactions. Alan Spivey,* Stellios Arseniyadis* Topics in Current Chemistry: Asymmetric Organocatalysis, Ed. B. List, Springer Verlag 2010, Vol 291, Chapter 25, pp 233280.

[23] Straightforward synthesis of the near-infrared fluorescent voltage-sensitive dye RH1691 and analogues thereof. Raphaël Lebeuf, Isabelle Férézou, Jean Rossier,Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2009, 11, 48224825.

[22] Enantioselective organocatalytic conjugate reduction of b-azole a,b-unsaturated aldehydes. Thomas J. Hoffman, Jyotirmayee Dash, James H. Rigby, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2009, 11, 27562759.

[21] One-pot hydrosilylation/RCM/protodesilylation: Application to the synthesis of w-alkenyl a,b-unsaturated lactones. Cyril Bressy, Frédéric Barggigia, Mathieu Guyonnet, Stellios Arseniyadis, Janine Cossy* Synlett, 2009, 565568.

[20] Asymmetric pentenylation of aldehydes: A new benchmark for the preparation of ethyl-substituted homoallylic alcohols. Ravindra P. Sonawane, Shyamsunder R. Joolakanti, Stellios Arseniyadis,* Janine Cossy* Synlett 2009, 213216.

[19] Asymmetric total synthesis of the immunosuppressant (-)-pironetin. Cyril Bressy, Jean-Pierre Vors, Stefan Hillebrand, Stellios Arseniyadis, Janine Cossy* Angew. Chem, Int. Ed. 2008, 47, 1013710140.

[18] Formal synthesis of leustroducsin B. Joëlle Moïse, Ravindra P. Sonawane, Camilla Corsi, Sebastian V. Wendeborn, Stellios Arseniyadis,* Janine Cossy* Synlett 2008, 26172620.

[17] Total synthesis of cystothiazole A by microwave-assisted olefin cross-metathesis. Julian Gebauer, Stellios Arseniyadis,* Janine Cossy* Eur. J. Org. Chem. 2008, 27012704.

[16] Synthesis of vinyl-functionalized oxazoles by olefin cross-metathesis. Thomas J. Hoffman, James H. Rigby, Stellios Arseniyadis, Janine Cossy* J. Org. Chem. 2008, 73, 24002403.

[15] Facile synthesis of the C1–C13 fragment of lyngbouilloside. Julian Gebauer, Stellios Arseniyadis,* Janine Cossy* Synlett 2008, 712714.

[14] Non-enzymatic kinetic resolution of amines in ionic liquids. Cyrille Sabot, Pithani V. Subhash, Alain Valleix, Stellios Arseniyadis,* Charles Mioskowski,* Synlett 2008, 268272.

[13] Chemical synthesis of a highly potent epothilone. Kyriakos C. Nicolaou, Benjamin Pratt, Stellios Arseniyadis (International publication number: WO2007062288A2, International publication date: 31/05/2007).

[12] A concise total synthesis of melithiazole C. Julian Gebauer, Stellios Arseniyadis, Janine Cossy* Org. Lett. 2007, 9, 34253427.

[11] The chemistry and biology of epothilones – The wheel keeps turning. Karl-Heinz Altmann,* Bernhard Pfeiffer, Stellios Arseniyadis, Benjamin A. Pratt, K. C. Nicolaou* ChemMedChem 2007, 396423.

[10] Cross-Metathesis between a-methylene-g-butyrolactone and olefins: A dramatic additive effect. Joëlle Moïse, Stellios Arseniyadis,* Janine Cossy* Org. Lett. 2007, 9, 16951698.

[9] Synthesis of vinyl-functionalized thiazoles by cross-metathesis and tandem Stille coupling/cross-metathesis. Jyotirmayee Dash, Stellios Arseniyadis, Janine Cossy* Adv. Synth. Cat. 2007, 349, 152156.

[8] Molecular design and chemical synthesis of a highly potent epothilone. K. C. Nicolaou,* Benjamin A. Pratt, Stellios Arseniyadis, Markus Wartmann, Aurora O’Brate, Paraskevi Giannakakou ChemMedChem 2006, 1, 4144.

[7] Rapid, room-temperature acylative kinetic resolution of sec-alcohols using atropisomeric 4-aminopyridine/triphenylphosphine catalysis. Alan C. Spivey,* Stellios Arseniyadis, Tomasz Fekner, Adrian Maddaford, David P. Leese Tetrahedron 2006, 62, 295301.

[6] Unprecedented, fully recyclable, solid-supported reagent for the kinetic resolution of racemic amines through enantioselective N-acetylation. Stellios Arseniyadis, Pithani V. Subhash, Alain Valleix, Alain Wagner,* Charles Mioskowski* Chem. Commun. 2005, 26, 33103312 (Highlighted in Synfacts 2005, 1, 170).

[5] Tuning the enantioselective N-acetylation of racemic amines: A spectacular salt effect. Stellios Arseniyadis, Pithani V. Subhash, Alain Valleix, Suju P. Mathew,Donna G. Blackmond, Alain Wagner,* Charles Mioskowski* J. Am. Chem. Soc. 2005, 127, 61386139.

[4] Nucleophilic catalysis by 4-(dialkylamino)pyridines revisited - The search for optimal reactivity and selectivity. Alan C. Spivey,* Stellios Arseniyadis Angew. Chem. Int. Ed. 2004, 43, 54365441.

[3] Kinetic resolution of amines: A chemoselective and highly enantioselective acetylating agent with a unique solvent-induced reversal of stereoselectivity. Stellios Arseniyadis, Alain Valleix, Alain Wagner,* Charles Mioskowski* Angew. Chem. Int. Ed. 2004, 43, 33143317.

[2] Resin bound 4-phenyl-1,2-dihydroquinoline (DHQ): An new safety-catch linker for solid phase organic synthesis (SPOS). Stellios Arseniyadis, Alain Wagner,* Charles Mioskowski* Tetrahedron Lett. 2004, 45, 22512253.

[1] A straightforward preparation of amino-polystyrene resin from Merrifield resin. Stellios Arseniyadis, Alain Wagner,* Charles Mioskowski* Tetrahedron Lett. 2002, 43, 97179719.


[2] Palladium precatalyst embodiments for enantioselective chemical reactions and methods of making and using the same. D. Leitch, S. Arseniyadis, J. Huang (International publication number: WO2023156972A1, International publication date: 24/08/2023).

[1] Chemical synthesis of a highly potent epothilone. Nicolaou, K. C.; Pratt, B.; Arseniyadis, S. (International publication number: WO2007062288, International publication date: 31/05/2007).